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About

Enable Innovative Drug Discover with DEL, FBDD and SBDD

  1. About
  2. Publications

Publications

  • 18 June 2020
    A Simple Method for Determining Compound Affinity and Chemical Yield From DNA-encoded Library Selections
    Biochemical and Biophysical Research Communications Volume 527, Issue 1, 18 June 2020, Pages 250-256
  • 27 April 2020
    Optimized Methods for IL-17A Refolding and anti-IL17A Fab Production for Co-Crystallization With Small Molecules
    BIOTECHNIQUESVOL. 69, NO. 1 https://doi.org/10.2144/btn-2019-0170
  • 10 April 2020
    Characterization of Specific N-α-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library
    ACS Med. Chem. Lett. 2020, 11, 6, 1175–1184 https://doi.org/10.1021/acsmedchemlett.0c00029
  • 02 April 2020
    Photocatalytic [2 + 2] Cycloaddition in DNA-Encoded Chemistry
    Org. Lett. 2020, 22, 8, 2908–2913 https://doi.org/10.1021/acs.orglett.0c00574
  • 12 February 2020
    RASS‐Enabled S/P−C and S−N Bond Formation for DEL Synthesis
    Angew. Chem. Int. Ed. 2020, 59, 7377 https://doi.org/10.1002/anie.201915493
  • 30 January 2020
    Synthesis of Multifunctional 2-Aminobenzimidazoles on DNA via Iodine-Promoted Cyclization
    Org. Lett. 2020, 22, 4, 1290–1294 https://doi.org/10.1021/acs.orglett.9b04578
  • 20 December 2019
    Exploring the Lower Limit of Individual DNA-Encoded Library Molecules in Selection
    SLAS Discov., 2019, 25, 5, 523-529 DOI: 10.1177/2472555219893949
  • 14 August 2019
    Synthesis of C3-Alkylated Indoles on DNA via Indolyl Alcohol Formation Followed by Metal-Free Transfer Hydrogenation
    Org. Lett. 2019, 21, 17, 6633–6637 https://doi.org/10.1021/acs.orglett.9b02132
  • 21 June 2019
    On-DNA Decarboxylative Arylation: Merging Photoredox with Nickel Catalysis in Water
    ACS Comb. Sci. 2019, 21, 8, 588–597 https://doi.org/10.1021/acscombsci.9b00076

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